Molecule Details
InChIKeyVYIKAHZTFTUSJO-UHFFFAOYSA-N
Compound NameN-[4-(3-Amino-1H-pyrazolo[3,4-d]pyrimidin-6-yl)-phenyl]-5-chloro-2-cyano-benzenesulfonamide
Canonical SMILESN#Cc1ccc(Cl)cc1S(=O)(=O)Nc1ccc(-c2ncc3c(N)n[nH]c3n2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.63
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O00141 SGK1 Homo sapiens Human PF00069 PF00433 8.5 IC50 ChEMBL;BindingDB
Q9HBY8 SGK2 Homo sapiens Human PF00069 PF00433 7.7 IC50 ChEMBL;BindingDB
Q96BR1 SGK3 Homo sapiens Human PF00069 PF00433 PF00787 6.7 IC50 ChEMBL;BindingDB