Molecule Details
InChIKeyVYHCLYDDXNTHAU-UHFFFAOYSA-N
Compound Name2-Azetidin-3-yl-8-bromo[1]benzofuro[3,2-d]pyrimidin-4(3H)-one
Canonical SMILESO=c1[nH]c(C2CNC2)nc2c1oc1ccc(Br)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL7.65
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
O00311 CDC7 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
P67870 CSNK2B Homo sapiens Human PF01214 7.4 IC50 ChEMBL
P68400 CSNK2A1 Homo sapiens Human PF00069 7.4 IC50 ChEMBL