Molecule Details
InChIKeyVXTOUZSUPQQPPE-UHFFFAOYSA-N
Compound NameN-[2-(1-benzylpiperidin-4-yl)ethyl]-5,6-dihydrobenzo[h]cinnolin-3-amine
Canonical SMILESc1ccc(CN2CCC(CCNc3cc4c(nn3)-c3ccccc3CC4)CC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.63
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P22303 ACHE Homo sapiens Human PF08674 PF00135 6.7 IC50 ChEMBL;BindingDB
P06276 BCHE Homo sapiens Human PF08674 PF00135 6.5 IC50 ChEMBL;BindingDB