Molecule Details
InChIKeyVXPAUBYOSZRWFR-DHZHZOJOSA-N
Compound Name4-[2-(4-Fluoro-phenyl)-propenyl]-2,6-dimethyl-phenol
Canonical SMILESC/C(=C\c1cc(C)c(O)c(C)c1)c1ccc(F)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.26
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P09917 ALOX5 Homo sapiens Human PF00305 PF01477 6.4 IC50 ChEMBL;BindingDB
P23219 PTGS1 Homo sapiens Human PF03098 6.2 IC50 ChEMBL
P35354 PTGS2 Homo sapiens Human PF03098 6.2 IC50 ChEMBL;BindingDB