Molecule Details
InChIKeyVXNXKGJSGMZXLZ-UHFFFAOYSA-N
Compound Name2-Methyl-5-(4-((4-sulfamoylphenyl)amino)phthalazin-1-yl)benzenesulfonamide
Canonical SMILESCc1ccc(-c2nnc(Nc3ccc(S(N)(=O)=O)cc3)c3ccccc23)cc1S(N)(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.62
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16790 CA9 Homo sapiens Human PF00194 9.3 IC50 ChEMBL;BindingDB
O14638 ENPP3 Homo sapiens Human PF01663 PF01033 7.3 Ki ChEMBL
P00918 CA2 Homo sapiens Human PF00194 6.3 IC50 ChEMBL;BindingDB