Molecule Details
InChIKeyVXKAOEFNKQZVOS-UHFFFAOYSA-N
Compound Name2-[3-[6-methyl-4-[4-(1H-pyrazol-4-yl)anilino]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]phenoxy]-N-pentan-3-ylacetamide
Canonical SMILESCCC(CC)NC(=O)COc1cccc(-c2nc3c(c(Nc4ccc(-c5cn[nH]c5)cc4)n2)CN(C)CC3)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.53
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11169 SLC2A3 Homo sapiens Human PF00083 6.2 IC50 ChEMBL;BindingDB
P11166 SLC2A1 Homo sapiens Human PF00083 6.1 IC50 ChEMBL;BindingDB
O97467 ht1 Plasmodium falciparum Pathogen PF00083 7.3 IC50 ChEMBL;BindingDB