Molecule Details
InChIKeyVWQADHAJYDYFRH-HCJIVJCNSA-O
Compound NameBz(4-tBu)-Phe-Ala-Leu-Lys(Me3)-Ser-OMe
Canonical SMILESCOC(=O)[C@H](CO)NC(=O)[C@H](CCCC[N+](C)(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc(C(C)(C)C)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.18
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O95931 CBX7 Homo sapiens Human PF17218 PF00385 7.5 IC50 ChEMBL;BindingDB
O00257 CBX4 Homo sapiens Human PF17218 PF00385 7.1 IC50 ChEMBL;BindingDB
Q8N8U2 CDYL2 Homo sapiens Human PF00385 PF00378 7.0 IC50 ChEMBL;BindingDB