6-(3,5-dimethyl-1,2-oxazol-4-yl)-2,2,4,4-tetramethyl-1H-quinolin-3-one

InChIKey	`VWCZQZNHWPQZGT-UHFFFAOYSA-N`
Compound Name	6-(3,5-dimethyl-1,2-oxazol-4-yl)-2,2,4,4-tetramethyl-1H-quinolin-3-one
Canonical SMILES	`Cc1noc(C)c1-c1ccc2c(c1)C(C)(C)C(=O)C(C)(C)N2`
Clinical Status	Data-mined Candidate
Targets (Human+Pathogen)	3
Pfam Stratification	Homologous
Avg pChEMBL	7.25
Source	ChEMBL;BindingDB

2D Structure

Activity Profile

Target	Gene	Organism	Category	Pfam	pChEMBL	Type	Source
P06401	PGR	Homo sapiens	Human	PF00104 PF02161 PF00105	7.7	Ki	ChEMBL;BindingDB
P04150	NR3C1	Homo sapiens	Human	PF02155 PF00104 PF00105	7.6	IC50	ChEMBL;BindingDB
P08235	NR3C2	Homo sapiens	Human	PF00104 PF00105	6.5	Ki	ChEMBL;BindingDB