Molecule Details
InChIKeyVVZPRTIRPLMIAE-RQBKSZSXSA-N
Compound Name(2S)-2-amino-N-[(3S,9R,14R,20S)-14-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]-3,20-dibenzyl-10,10,13,13-tetramethyl-2,5,8,15,18,21-hexaoxo-11,12-dithia-1,4,7,16,19,22-hexazabicyclo[20.2.2]hexacosan-9-yl]-3-(4-hydroxyphenyl)propanamide
Canonical SMILESCC1(C)SSC(C)(C)[C@H](NC(=O)[C@@H](N)Cc2ccc(O)cc2)C(=O)NCC(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCN(CC2)C(=O)[C@H](Cc2ccccc2)NC(=O)CNC(=O)[C@H]1NC(=O)[C@@H](N)Cc1ccc(O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.5
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41143 OPRD1 Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB