Molecule Details
InChIKeyVVRNZKKUOWFMOX-NRWPOFLRSA-N
Compound NameN-[(4R)-1-(1-acetylpiperidine-4-carbonyl)-3-(3,4-dichlorophenyl)piperidin-4-yl]-4-bromo-N-methylbenzamide
Canonical SMILESCC(=O)N1CCC(C(=O)N2CC[C@@H](N(C)C(=O)c3ccc(Br)cc3)C(c3ccc(Cl)c(Cl)c3)C2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.05
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21452 TACR2 Homo sapiens Human PF00001 9.3 IC50 ChEMBL;BindingDB
Q9UHF0 TAC3 Homo sapiens Human PF03823 7.6 IC50 ChEMBL;BindingDB
P25103 TACR1 Homo sapiens Human PF00001 7.2 IC50 ChEMBL;BindingDB