Molecule Details
InChIKeyVVOQENFAZBJUSR-NDEPHWFRSA-N
Compound Name(S)-1-methyl-N-(1-(5-(naphthalen-2-yl)-1H-imidazol-2-yl)-7-oxoundecyl)piperidine-4-carboxamide
Canonical SMILESCCCCC(=O)CCCCC[C@H](NC(=O)C1CCN(C)CC1)c1ncc(-c2ccc3ccccc3c2)[nH]1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.0
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q02161 RHD Homo sapiens Human PF00909 7.1 pIC50 TTD_MultiTarget
Q13547 HDAC1 Homo sapiens Human PF00850 7.1 pIC50 TTD_MultiTarget
O15379 HDAC3 Homo sapiens Human PF00850 6.7 IC50 ChEMBL;BindingDB