Molecule Details
InChIKeyVVNAQHKXBHSZIX-WIPVZAJSSA-N
Compound NameAc-D-Asp(1)-D-His-Phe-D-Arg-Trp-D-Ala-D-Lys(1)-NH2
Canonical SMILESCC(=O)N[C@@H]1CC(=O)NCCCC[C@H](C(N)=O)NC(=O)[C@@H](C)NC(=O)[C@H](Cc2c[nH]c3ccccc23)NC(=O)[C@@H](CCCN=C(N)N)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](Cc2c[nH]cn2)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.14
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q01726 MC1R Homo sapiens Human PF00001 8.7 IC50 ChEMBL;BindingDB
P32245 MC4R Homo sapiens Human PF00001 8.7 IC50 ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 7.0 IC50 ChEMBL;BindingDB