Molecule Details
InChIKeyVTXMFBVROQUZNI-UHFFFAOYSA-N
Compound Name1-(6-(Aminomethyl)-5-(2,4-dichlorophenyl)-7-methylimidazo[1,2-a]pyrimidin-2-yl)-2-(pyridin-3-ylamino)ethanone
Canonical SMILESCc1nc2nc(C(=O)N(C)Cc3cccnc3)cn2c(-c2ccc(Cl)cc2Cl)c1CN
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q6V1X1 DPP8 Homo sapiens Human PF19520 PF00930 PF00326 9.4 Ki ChEMBL;BindingDB
Q86TI2 DPP9 Homo sapiens Human PF19520 PF00930 PF00326 9.2 Ki ChEMBL;BindingDB
P27487 DPP4 Homo sapiens Human PF00930 PF00326 8.6 Ki ChEMBL;BindingDB