Molecule Details
InChIKeyVTWJQIYQJKMCSP-UHFFFAOYSA-N
Compound Name3-ethyl-8-[1-[[5-oxo-1-[4-(trifluoromethyl)phenyl]pyrrolidin-3-yl]methyl]pyrazol-4-yl]-1-propyl-7H-purine-2,6-dione
Canonical SMILESCCCn1c(=O)c2[nH]c(-c3cnn(CC4CC(=O)N(c5ccc(C(F)(F)F)cc5)C4)c3)nc2n(CC)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29275 ADORA2B Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB