Molecule Details
InChIKeyVTRPSKIFOIGMRA-UHFFFAOYSA-N
Compound Name2-fluoro-6-[(2-{[1-(1H-imidazol-1-ylacetyl)-5-(methyloxy)-2,3-dihydro-1H-indol-6-yl]amino}-1H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]benzamide
Canonical SMILESCOc1cc2c(cc1Nc1nc(Nc3cccc(F)c3C(N)=O)c3cc[nH]c3n1)N(C(=O)Cn1ccnc1)CC2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.06
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08069 IGF1R Homo sapiens Human PF00757 PF07714 PF01030 7.5 IC50 ChEMBL;BindingDB
P06729 CD2 Homo sapiens Human PF05790 PF07686 7.5 pIC50 TTD_MultiTarget
P45983 MAPK8 Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB