Molecule Details
InChIKeyVTQSIRZSABRYHH-SZPZYZBQSA-N
Compound Namecis-6-(3,5-Dimethylpiperazin-1-yl)-5-methoxy-1-[4-(6-methylpyridin-2-yl)-1-naphthoyl]indoline
Canonical SMILESCOc1cc2c(cc1N1C[C@@H](C)N[C@@H](C)C1)N(C(=O)c1ccc(-c3cccc(C)n3)c3ccccc13)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.73
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28222 HTR1B Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB
P28221 HTR1D Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.0 Ki ChEMBL;BindingDB