Molecule Details
InChIKeyVTGUKXAQUOKKSW-UHFFFAOYSA-N
Compound Name5-Amino-3-(1,3-benzothiazol-5-yl)-1-ethylpyrazole-4-carboxamide
Canonical SMILESCCn1nc(-c2ccc3scnc3c2)c(C(N)=O)c1N
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.41
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43353 RIPK2 Homo sapiens Human PF00619 PF07714 6.7 IC50 ChEMBL;BindingDB
P36897 TGFBR1 Homo sapiens Human PF01064 PF00069 PF08515 6.5 IC50 ChEMBL;BindingDB
P06239 LCK Homo sapiens Human PF07714 PF00017 PF00018 6.0 IC50 ChEMBL;BindingDB