Molecule Details
InChIKeyVTEVEQHENPPCQK-UHFFFAOYSA-N
Canonical SMILESCc1ccccc1CN(Cc1cc(=O)[nH]c2c(F)c(F)ccc12)c1cnccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P35228 NOS2 Homo sapiens Human PF00667 PF00258 PF00175 PF02898 8.0 IC50 ChEMBL;BindingDB
P29475 NOS1 Homo sapiens Human PF00667 PF00258 PF00175 PF02898 PF00595 7.3 IC50 ChEMBL;BindingDB