Molecule Details
InChIKeyVTABFDXOHRLLHO-IHBRBHLJSA-N
Compound Name1-((S)-((S)-1-Carboxy-3-methyl-butylcarbamoyl)-{(S)-2-[(S)-2-(2-ethyl-butyrylamino)-3,3-dimethyl-butyrylamino]-4-oxo-4-pyrrolidin-1-yl-butyrylamino}-methyl)-cyclopent-3-enecarboxylic acid
Canonical SMILESCCC(CC)C(=O)N[C@H](C(=O)N[C@@H](CC(=O)N1CCCC1)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)O)C1(C(=O)O)CC=CC1)C(C)(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.19
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P23921 RRM1 Homo sapiens Human PF03477 PF02867 PF00317 8.2 IC50 ChEMBL;BindingDB
P31350 RRM2 Homo sapiens Human PF00268 8.2 IC50 ChEMBL
Q7LG56 RRM2B Homo sapiens Human PF00268 8.2 IC50 ChEMBL