Molecule Details
InChIKeyVTAARTQTOOYTES-RGDLXGNYSA-N
Compound Name(+)-2-Aminobicyclo(3.1.0)hexane-2,6-dicarboxylic acid
Canonical SMILESN[C@@]1(C(=O)O)CC[C@H]2[C@H](C(=O)O)[C@H]21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.08
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB21031
Drug NameEglumetad
CAS Number176199-48-7
Groups experimental
ATC Codes nan
DescriptionEglumetad is a small molecule drug. Eglumetad has a monoisotopic molecular weight of 185.07 Da.

Categories: Anti-Anxiety Agents Bridged-Ring Compounds Central Nervous System Agents Central Nervous System Depressants Excitatory Amino Acid Agents Excitatory Amino Acid Agonists Neurotransmitter Agents Psychotropic Drugs Tranquilizing Agents
Cross-references: BindingDB: 50397661 ChEBI: 194387 CHEMBL8759 PDB: 40F ZINC: ZINC000003824390
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q14416 GRM2 Homo sapiens Human PF00003 PF01094 PF07562 7.1 Ki ChEMBL;BindingDB
Q14832 GRM3 Homo sapiens Human PF00003 PF01094 PF07562 7.0 Ki ChEMBL;BindingDB
DrugBank Target Actions (2)
Target Gene Target Name Action Type
Q14416 GRM2 Metabotropic glutamate receptor 2 agonist targets
Q14832 GRM3 Metabotropic glutamate receptor 3 agonist targets