Molecule Details
InChIKeyVSSMWFPLHKIWCP-UHFFFAOYSA-N
Compound Name4-(3-Cyclopropyl-6-fluoroimidazo[1,2-a]pyridin-2-yl)isoquinoline
Canonical SMILESFc1ccc2nc(-c3cncc4ccccc34)c(C3CC3)n2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.49
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P19099 CYP11B2 Homo sapiens Human PF00067 9.3 IC50 ChEMBL;BindingDB
P15538 CYP11B1 Homo sapiens Human PF00067 7.1 IC50 ChEMBL;BindingDB
P11511 CYP19A1 Homo sapiens Human PF00067 6.1 IC50 ChEMBL;BindingDB