Molecule Details
InChIKeyVRUYMJKZIKNSKH-UHFFFAOYSA-N
Compound Name6-[(3-Chloro-4-cyano-phenyl)-(3-methyl-3H-imidazol-4-yl)-methoxymethyl]-1-methyl-2-oxo-5-(4-trifluoromethoxy-phenyl)-1,2-dihydro-pyridine-3-carbonitrile
Canonical SMILESCn1cncc1C(OCc1c(-c2ccc(OC(F)(F)F)cc2)cc(C#N)c(=O)n1C)c1ccc(C#N)c(Cl)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.57
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 9.4 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 9.4 IC50 ChEMBL
P53609 PGGT1B Homo sapiens Human PF00432 6.8 IC50 ChEMBL