Molecule Details
InChIKeyVRMQALIKUKOPIW-UHFFFAOYSA-N
Compound NameN-(4-fluorophenyl)-2-[4-oxo-3-[2-(4-sulfamoylphenyl)ethyl]quinazolin-2-yl]sulfanylacetamide
Canonical SMILESNS(=O)(=O)c1ccc(CCn2c(SCC(=O)Nc3ccc(F)cc3)nc3ccccc3c2=O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16790 CA9 Homo sapiens Human PF00194 7.9 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 7.6 Ki ChEMBL;BindingDB
P00915 CA1 Homo sapiens Human PF00194 7.5 Ki ChEMBL;BindingDB