Molecule Details
InChIKeyVRENQJJXDFBYMO-FAIXQHPJSA-N
Compound Name2-[4-[2-[3-[4-[4-[[2-[(2S)-2-(1,3-benzoxazole-2-carbonyl)pyrrolidin-1-yl]-2-oxoethyl]carbamoyl]quinolin-6-yl]phenyl]sulfonylpropylamino]-2-oxoethyl]-7,10-bis(carboxymethyl)-1,4,7,10-tetrazacyclododec-1-yl]acetic acid
Canonical SMILESO=C(O)CN1CCN(CC(=O)O)CCN(CC(=O)NCCCS(=O)(=O)c2ccc(-c3ccc4nccc(C(=O)NCC(=O)N5CCC[C@H]5C(=O)c5nc6ccccc6o5)c4c3)cc2)CCN(CC(=O)O)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.3
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5JRX3 PITRM1 Homo sapiens Human PF08367 PF00675 PF05193 PF22516 8.2 IC50 BindingDB
P27487 DPP4 Homo sapiens Human PF00930 PF00326 6.4 IC50 BindingDB