Molecule Details
InChIKeyVQNCHRIEHZHEQE-UHFFFAOYSA-N
Compound Name2,2,2-Trifluoro-1-[4-(4-fluoroanilino)pyrimidin-5-yl]-1-(1-methylsulfonylpiperidin-4-yl)ethanol
Canonical SMILESCS(=O)(=O)N1CCC(C(O)(c2cncnc2Nc2ccc(F)cc2)C(F)(F)F)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.55
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P15538 CYP11B1 Homo sapiens Human PF00067 8.7 IC50 ChEMBL;BindingDB
P19099 CYP11B2 Homo sapiens Human PF00067 8.4 IC50 ChEMBL;BindingDB