Molecule Details
InChIKeyVQLPLYSROCPWFF-QZTJIDSGSA-N
Compound Namerel-3,4-Dichloro-N-methyl-N-((1R,2R)-2-(1-pyrrolidinyl)cyclohexyl)benzeneacetamide
Canonical SMILESCN(C(=O)Cc1ccc(Cl)c(Cl)c1)[C@@H]1CCCC[C@H]1N1CCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL7.45
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P41145 OPRK1 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 8.6 IC50 BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 6.3 Ki BindingDB
Q99720 SIGMAR1 Homo sapiens Human PF04622 6.1 Ki BindingDB