Molecule Details
InChIKeyVQJKUVSKZOTZTB-UHFFFAOYSA-N
Compound Name4-[1-(2,6-difluorophenyl)ethyl]-2-[isopropyl(methyl)amino]-5-methyl-1H-pyrimidin-6-one
Canonical SMILESCc1c(C(C)c2c(F)cccc2F)nc(N(C)C(C)C)[nH]c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.43
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9WKE8 reverse transcriptase Human immunodeficiency virus type 1 Pathogen PF00078 7.5 Ki BindingDB
Q72547 pol Human immunodeficiency virus type 1 Pathogen PF00075 PF00078 PF06815 PF06817 7.4 Ki ChEMBL