Molecule Details
InChIKeyVQGGQIGYLGHRNK-UHFFFAOYSA-N
Compound Name2-(3-Anilino-2-methylquinoxalin-5-yl)-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-one
Canonical SMILESCc1nc2cccc(-c3cc4c([nH]3)CCNC4=O)c2nc1Nc1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.04
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 6.7 IC50 ChEMBL