Molecule Details
InChIKeyVQAHFLPDFJAHTG-UHFFFAOYSA-N
Compound Name9-cyclopentyl-8-N-(2,6-difluorophenyl)-2-N-(4-methoxyphenyl)purine-2,8-diamine
Canonical SMILESCOc1ccc(Nc2ncc3nc(Nc4c(F)cccc4F)n(C4CCCC4)c3n2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.12
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P45984 MAPK9 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB