Molecule Details
InChIKeyVOXOJYXJGWUWQI-UHFFFAOYSA-N
Compound Namemethyl 1-[3-[[4-(2,1,3-benzoxadiazol-5-yl)-2,5-dioxo-4,7-dihydro-1H-furo[3,4-d]pyrimidine-3-carbonyl]amino]propyl]-4-phenylpiperidine-4-carboxylate
Canonical SMILESCOC(=O)C1(c2ccccc2)CCN(CCCNC(=O)N2C(=O)NC3=C(C(=O)OC3)C2c2ccc3nonc3c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.35
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB