Molecule Details
InChIKeyVOFLAIHEELWYGO-UHFFFAOYSA-N
Canonical SMILESO=C(c1cc(Cl)c(O)c(Cl)c1)N1CS(=O)(=O)c2ccccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.43
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB16145
Drug NameDotinurad
CAS Number1285572-51-1
Groups investigational
ATC Codes nan
DescriptionDotinurad is under investigation in clinical trial NCT03372200 (Febuxostat-controlled, Double-blind, Comparative Study of FYU-981 in Hyperuricemia With or Without Gout).

Categories: Antigout Preparations Antirheumatic Agents Heterocyclic Compounds, Fused-Ring Thiazoles Uricosuric Agents
Cross-references: ChemSpider: 59718651 PDB: A1AIK
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96S37 SLC22A12 Homo sapiens Human PF07690 7.4 IC50 ChEMBL;BindingDB
Q9UNQ0 ABCG2 Homo sapiens Human PF01061 PF19055 PF00005 7.4 IC50 ChEMBL
DrugBank Target Actions (1)
Target Gene Target Name Action Type
Q96S37 SLC22A12 Solute carrier family 22 member 12 inhibitor targets