Molecule Details
InChIKeyVNXLMJGQXWEBFC-NWDGAFQWSA-N
Compound Name4-[(1S,2R)-2-(cyclopropylmethylamino)cyclopropyl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)thiophene-2-carboxamide
Canonical SMILESCc1nnc(NC(=O)c2cc([C@@H]3C[C@H]3NCC3CC3)cs2)s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.6
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O60341 KDM1A Homo sapiens Human PF01593 PF04433 6.6 IC50 ChEMBL;BindingDB
P09211 GSTP1 Homo sapiens Human PF14497 PF02798 6.6 IC50 BindingDB
Q9UKL0 RCOR1 Homo sapiens Human PF01448 PF00249 PF20878 6.6 IC50 ChEMBL