Molecule Details
InChIKeyVNGIYBDBGMQECO-UHFFFAOYSA-N
Compound Name6-(3-sulfamoyl-2-(2H-tetrazol-5-yl)phenyl)quinoline-2-carboxylic acid
Canonical SMILESNS(=O)(=O)c1cccc(-c2ccc3nc(C(=O)O)ccc3c2)c1-c1nn[nH]n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.8
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.1 IC50 ChEMBL;BindingDB
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 7.5 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 6.8 IC50 BindingDB