Molecule Details
InChIKeyVMUAYDSPKYLLJV-XLNRJJMWSA-N
Compound Name(Z)-N-[3-({3-[3-(Dimethylamino)propyl]-4-oxo-4,5,6,7-tetrahydro-1H-indol-2-yl}methylene)-2-oxoindolin-5-yl]benzenesulfonamide
Canonical SMILESCN(C)CCCc1c(/C=C2\C(=O)Nc3ccc(NS(=O)(=O)c4ccccc4)cc32)[nH]c2c1C(=O)CCC2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.32
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 6.6 IC50 ChEMBL
O75716 STK16 Homo sapiens Human PF00069 6.3 pIC50 TTD_MultiTarget
Q02161 RHD Homo sapiens Human PF00909 6.0 pIC50 TTD_MultiTarget