Molecule Details
InChIKeyVMOVOUMHZIMENS-UHFFFAOYSA-N
Compound Name6-(Phenothiazin-10-ylmethyl)pteridine-2,4-diamine
Canonical SMILESNc1nc(N)c2nc(CN3c4ccccc4Sc4ccccc43)cnc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O30463 folA Mycobacterium avium Pathogen PF00186 7.5 IC50 ChEMBL;BindingDB
Q07422 Toxoplasma gondii Pathogen PF00186 PF00303 7.0 IC50 ChEMBL;BindingDB