Molecule Details
InChIKeyVMHDSBUIYYCTCD-UHFFFAOYSA-N
Compound Name1-[N-[(4-cyanophenyl)methyl]-4-fluoroanilino]-3-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propyl]urea
Canonical SMILESCOc1ccccc1N1CCN(CCCNC(=O)NN(Cc2ccc(C#N)cc2)c2ccc(F)cc2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.94
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB