Molecule Details
InChIKeyVMGFMOIZZDBILY-DMBLRCPMSA-N
Compound Name2-[(S)-[[(2S)-2-[[(2S)-1-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-phenylmethyl]prop-2-enoic acid
Canonical SMILESC=C(C(=O)O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](N)Cc1c(C)cc(O)cc1C)c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35372 OPRM1 Homo sapiens Human PF00001 10.5 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 7.6 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB