Molecule Details
InChIKeyVLKJKVMACAESPP-BHHOHBANSA-N
Compound Name1-(3-(125I)iodophenyl)-3-[(3S)-1-methyl-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]urea
Canonical SMILESCN1C(=O)[C@@H](NC(=O)Nc2cccc([125I])c2)N=C(c2ccccc2)c2ccccc21
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.0
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 9.0 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 9.0 Ki ChEMBL