Molecule Details
InChIKeyVKZGOHFGTOOZHY-UHFFFAOYSA-N
Compound NameN-[5-(2-methoxyphenoxy)-6-[3-[(4-methylphenyl)sulfonylamino]propoxy]-2-morpholin-4-ylpyrimidin-4-yl]-5-propan-2-ylpyridine-2-sulfonamide
Canonical SMILESCOc1ccccc1Oc1c(NS(=O)(=O)c2ccc(C(C)C)cn2)nc(N2CCOCC2)nc1OCCCNS(=O)(=O)c1ccc(C)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.28
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24530 EDNRB Homo sapiens Human PF00001 7.6 IC50 ChEMBL;BindingDB
P25101 EDNRA Homo sapiens Human PF00001 6.9 IC50 ChEMBL;BindingDB