Molecule Details
InChIKeyVKWYVNKUABAQRG-ABRORHJPSA-N
Compound Name(1S,16R)-13-(cyclopropylmethyl)-1,16-dimethyl-5,6,7,13-tetraazatetracyclo[10.3.1.0^{2,10}.0^{4,8}]hexadeca-2,4(8),6,9-tetraene
Canonical SMILESC[C@H]1C2Cc3cc4nn[nH]c4cc3[C@@]1(C)CCN2CC1CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.13
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41145 OPRK1 Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB