Molecule Details
InChIKeyVKTSBOIQJNMQAL-UHFFFAOYSA-N
Canonical SMILESCC(=O)Nc1cc(-c2ccc(N3CCN(C(=O)c4cc(Cc5n[nH]c(=O)c6ccccc56)ccc4F)CC3)nc2)cc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c1C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.89
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96NZ9 PRAP1 Homo sapiens Human PF15314 8.2 IC50 ChEMBL;BindingDB
Q15910 EZH2 Homo sapiens Human PF21358 PF11616 PF18118 PF18264 PF00856 7.6 IC50 ChEMBL;BindingDB