Molecule Details
InChIKeyVKTAENBLRPMXKK-UHFFFAOYSA-N
Compound Name3-(6-(2-chlorophenylamino)-1H-indazol-3-yl)-N-(piperidin-4-yl)benzamide
Canonical SMILESO=C(NC1CCNCC1)c1cccc(-c2n[nH]c3cc(Nc4ccccc4Cl)ccc23)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.13
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 8.9 IC50 ChEMBL;BindingDB
Q16539 MAPK14 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB