Molecule Details
InChIKeyVKCYYRCBSOAUCN-UHFFFAOYSA-N
Compound Name3,4,5-trimethoxy-N-(5-sulfamoyl-1,3,4-thiadiazol-2-yl)benzamide
Canonical SMILESCOc1cc(C(=O)Nc2nnc(S(N)(=O)=O)s2)cc(OC)c1OC
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.35
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 8.0 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.0 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 6.0 Ki ChEMBL;BindingDB