Molecule Details
InChIKeyVJXUXTWQBIILQL-CQSZACIVSA-N
Compound Name(R)-3-amino-N-(5-(3-(aminomethyl)piperidin-1-yl)-1-methyl-1H-pyrazol-4-yl)-6-(2-fluorophenyl)picolinamide
Canonical SMILESCn1ncc(NC(=O)c2nc(-c3ccccc3F)ccc2N)c1N1CCC[C@H](CN)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.78
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.5 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 8.9 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.0 Ki ChEMBL;BindingDB