Molecule Details
InChIKeyVJUQIMXHRMEYAS-UHFFFAOYSA-N
Compound Name8-hydroxy-5-[4-[4-[(2-oxo-3,4-dihydro-1H-quinolin-7-yl)oxy]butyl]piperazin-1-yl]-1H-quinolin-2-one
Canonical SMILESO=C1CCc2ccc(OCCCCN3CCN(c4ccc(O)c5[nH]c(=O)ccc45)CC3)cc2N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.04
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 7.9 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB