Molecule Details
InChIKeyVJAAXPKEDHFXAO-UHFFFAOYSA-N
Compound Name1-[3-Chloro-4-(4-methylpiperazin-1-yl)sulfonylphenyl]-5-[2-ethoxy-5-(4-methylpiperazin-1-yl)sulfonylphenyl]-3-methylpyrazolo[4,5-e][1,2,4]triazine
Canonical SMILESCCOc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1-c1nnc2c(n1)c(C)nn2-c1ccc(S(=O)(=O)N2CCN(C)CC2)c(Cl)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43570 CA12 Homo sapiens Human PF00194 7.1 Ki ChEMBL;BindingDB
Q16790 CA9 Homo sapiens Human PF00194 6.4 Ki ChEMBL;BindingDB
P00915 CA1 Homo sapiens Human PF00194 6.2 Ki ChEMBL;BindingDB