Molecule Details
InChIKeyVITDWMDDGMNHHH-UHFFFAOYSA-N
Compound Name1-(3-{[5-Carbamoyl-4-methyl-6-(4-nitro-phenyl)-2-oxo-3,6-dihydro-2H-pyrimidine-1-carbonyl]-amino}-propyl)-4-phenyl-piperidine-4-carboxylic acid methyl ester
Canonical SMILESCOC(=O)C1(c2ccccc2)CCN(CCCNC(=O)N2C(=O)NC(C)=C(C(N)=O)C2c2ccc([N+](=O)[O-])cc2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 9.2 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB