Molecule Details
InChIKeyVINQLWACVZJJIO-UHFFFAOYSA-N
Compound NameN-(4-cyano-3-(1H-1,2,4-triazol-5-yl)thiophen-2-yl)-2-(isoquinolin-5-yl)acetamide
Canonical SMILESN#Cc1csc(NC(=O)Cc2cccc3cnccc23)c1-c1ncn[nH]1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.9
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB