Molecule Details
InChIKeyVIESBBSLVITZSP-UHFFFAOYSA-N
Compound Name3-[[5-[5-(6-chloro-1H-benzimidazol-2-yl)-2-pyridinyl]-2-pyridinyl]oxy]-2,2-dimethylpropanoic acid
Canonical SMILESCC(C)(COc1ccc(-c2ccc(-c3nc4cc(Cl)ccc4[nH]3)cn2)cn1)C(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.58
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O75907 DGAT1 Homo sapiens Human PF03062 9.2 IC50 ChEMBL;BindingDB
P35610 SOAT1 Homo sapiens Human PF03062 6.0 IC50 ChEMBL;BindingDB