Molecule Details
InChIKeyVHZVQRFYYPOCQY-JTQLQIEISA-N
Compound Name(S)-1-(4-Sulfamoyl-phenylthiocarbamoyl)-pyrrolidine-2-carboxylic acid
Canonical SMILESNS(=O)(=O)c1ccc(NC(=S)N2CCC[C@H]2C(=O)O)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.39
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 7.6 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.6 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 7.0 Ki ChEMBL;BindingDB